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Fluoxetine Hydrochloride Orodispersible Tablets; Formulation, Taste masking, Evaluation, Stability and In vivo studies

Article

Last updated: 13 Dec 2022

Subjects

-

Tags

Fluoxetine HCl, &beta
-cyclodextrin, Superdisintegrants, Stability, In vivo study
Fluoxetine Hydrochloride Orodispersible Tablets; Formulation, Taste masking, Evaluation, Stability and In vivo studies
The 1st International Online Conference Pharmaceutical and Medical Sciences: A Response to COVID-19 Theme: Support Healthcare Heroes
Pharmaceutical revolution

Abstract

The purpose was to design and evaluate Fluoxetine orodispersible tablets (FLX ODTs) that characterized by, fast drug release with acceptable taste. FLX ODTs were prepared by direct compression after complexation of FLX with β-cyclodextrin (β-CD) for taste masking, using Crospovidone (CP), croscarmellose sodium (Ac-di-sol), sodium starch glycolate (SSG) and indion (as superdisintegrants). The powder blend was evaluated for pre-compression parameters. Also, the prepared tablets were evaluated for post-compression parameters. The selected tablet formulations based upon drug release at 40 sec and acceptable release pattern were investigated for accelerated stability testing and for comparative in vivo study with a marketed product. Results showed that all powder blends had good flow properties and all the prepared tablets complied with the pharmacopeial requirements for uniformity of content, weight, friability, and hardness. Also, all the tablets acquired acceptable taste after complexation. Order of release of the drug, regarding superdisintegrants used, was as in the following descending order: CP> Ac-di-sol> SSG> indion. Accelerated stability study of selected formulation F2 and F6 showed that; there was no considerable change in physical properties, drug content and percentage drug release, also the in vivo study proved the effectiveness of FLX ODTs as anti-depressant. The results obtained showed a promising potential of ODTs containing a specific ratio of superdisintegrants and prepared by complexation method for the effective treatment of depression.

Categories

Pharmaceutical revolution

Keywords

Fluoxetine HCl, &beta, -cyclodextrin, Superdisintegrants, Stability, In vivo study

Authors

First Name

Dina

Last Name

Osman

Affiliation

pharmaceutics and industrial pharmacy, Faculty of pharmacy, al Azhar Uni, cairo,egypt

Email

-

City

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Orcid

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First Name

Maha

Last Name

Marzouk

Affiliation

Pharmaceutics and industrial pharmacy, Faculty of pharmacy(girls), al Azhar Uni, cairo, egypt

Email

-

City

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Orcid

-

First Name

omnia

Last Name

mohamed

Affiliation

pharmaceutics and industrial pharmacy, Faculty of pharmacy(girls), al Azhar Uni, cairo, egypt

Email

-

City

-

Orcid

-

Publish Date

14 Jun 2021

Link

https://pmsazhar.conferences.ekb.eg/article_1107.html

Order

60

Publication Type

Conference

Publication Title

The 1st International Online Conference Pharmaceutical and Medical Sciences: A Response to COVID-19 Theme: Support Healthcare Heroes

Publication Link

https://pmsazhar.conferences.ekb.eg/

Details

Type

Article

Locale

en

Created At

13 Dec 2022