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169358

SUSTAINED RELEASE BEHAVIOR OF FAMOTIDINE FROM FLOATING GELUCIRE FORMULATIONS

Article

Last updated: 22 Jan 2023

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Abstract

The aim of the present study was to prepare floating sustained release formulations of famotidine (FM) using a blend of Gelucire 43/01 (GL 43/01) and Gelucire 44/14 (GL 44/14) in different concentrations. These formulations were intended to be retained in the stomach and prolong the drug release to improve bioavailability and reduce frequency of administration. Granules and beads were prepared by melt-granulation technique and melt-solidification technique, respectively. The formulations were evaluated for surface morphology, flowability, in-vitro floating ability, and in-vitro drug release. In case of beads, process yield, drug loading, encapsulation efficiency, and particle size were also investigated. Differential scanning calorimetry (DSC) and infrared spectroscopy (IR) were used to investigate the possibility of drug-lipid interactions. The obtained beads had smooth surfaces, while the granules showed rough surfaces. Both formulations showed free flowing properties and excellent floating characteristics. There was no interaction between the drug and Gelucires used in the formulation. In-vitro drug release of FM from the prepared granules and beads was studied in 0.1 N HCI (pH 1.2) for up to 12 hrs. The drug released in a sustained manner in pH 1.2 from both formulations with no significant difference between granules and beads.

DOI

10.21608/zjps.2009.169358

Authors

First Name

Gihan

Last Name

Fetih

MiddleName

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Affiliation

Department of Pharmaceutics, Faculty of Pharmacy, Assiut University, Assiut, Egypt

Email

gihan.fetih@yahoo.com

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Orcid

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Volume

18

Article Issue

2

Related Issue

23549

Issue Date

2009-12-01

Receive Date

2009-09-28

Publish Date

2009-12-01

Page Start

16

Page End

25

Print ISSN

1110-5089

Online ISSN

2356-9786

Link

https://zjps.journals.ekb.eg/article_169358.html

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https://zjps.journals.ekb.eg/service?article_code=169358

Order

3

Type

Original Article

Type Code

862

Publication Type

Journal

Publication Title

Zagazig Journal of Pharmaceutical Sciences

Publication Link

https://zjps.journals.ekb.eg/

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Article

Created At

22 Jan 2023