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7187

UTILITIES OF CYANOTHIOFORMAMIDES AND IMIDAZOLIDINEIMINO-THIONES IN THE SYNTHESIS OF NEW TYPES OF OXADIAZOLE, TRIAZOLTHIONE, BENZOTHIAZOLOQUINAZOLINONE, PYRROLO[2,3-B] PYRROLE AND

Article

Last updated: 03 Jan 2025

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Chemistry

Abstract

Cyanothioformamides were reacted with benzoyl hydrazine, acetyl hydrazine and anthranilic acid to afford oxadiazole (4), triazolthione (5) and benzothiazoloquinazolinone derivatives (6) respectively. They also reacted with thiocarbohydrazide, semicarbazide, thiosemicarbazide and active methylene compounds to produce 3-hydrazino-1,2-,4-triazol-5-thione (8), thiocarbamoylsemicarbazide (9), triazolidinedithione (10). Treatment of imidazolidine iminothiones with different nucleophilic reagents gave imidazotriazines besides other imidazolidine derivatives. Some of the newly synthestized derivatives were screened for antibacterial and antifungal activity and showed prononced antimicrobial activity.

DOI

10.21608/absb.2011.7187

Keywords

CYANOTHIOFORMAMIDES, IMIDAZOLIDINEIMINO-THIONES, Oxadiazole, TRIAZOLTHIONE

Authors

First Name

F.

Last Name

MAHMOUD

MiddleName

F.

Affiliation

Chemistry Department, Faculty of Science, Al-Azhar University (for Girls), Cairo, Egypt

Email

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Orcid

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First Name

N.

Last Name

TAHA

MiddleName

M.

Affiliation

Chemistry Department, Faculty of Science, Al-Azhar University (for Girls), Cairo, Egypt

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-

City

-

Orcid

-

First Name

A.

Last Name

EL-SHARIEF

MiddleName

M.

Affiliation

Chemistry Department, Faculty of Science, Al-Azhar University (for Boys), Cairo, Egypt

Email

-

City

-

Orcid

-

First Name

E.

Last Name

AHMED

MiddleName

M.

Affiliation

Chemistry Department, Faculty of Science, Al-Azhar University (for Girls), Cairo, Egypt

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-

City

-

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-

Volume

22

Article Issue

Issue 1-A

Related Issue

1363

Issue Date

2011-06-01

Receive Date

2011-01-02

Publish Date

2011-06-01

Page Start

163

Page End

186

Print ISSN

1110-2535

Online ISSN

2636-3305

Article File

ABSB_Volume 22_Issue Issue 1-A_Pages 163-186.pdf

PDF . 363.4kB

Link

https://absb.journals.ekb.eg/article_7187.html

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https://absb.journals.ekb.eg/service?article_code=7187

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12

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Original Article

Type Code

520

Publication Type

Journal

Publication Title

Al-Azhar Bulletin of Science

Publication Link

https://absb.journals.ekb.eg/

MainTitle

UTILITIES OF CYANOTHIOFORMAMIDES AND IMIDAZOLIDINEIMINO-THIONES IN THE SYNTHESIS OF NEW TYPES OF OXADIAZOLE, TRIAZOLTHIONE, BENZOTHIAZOLOQUINAZOLINONE, PYRROLO[2,3-B] PYRROLE AND IMIDAZOTRIAZINE DERIVATIVES OF BIOLOGICAL INTEREST.

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Article

Created At

22 Jan 2023